Association of ABCB1, CYP3A4*18B and CYP3A5*3 genotypes with the pharmacokinetics of tacrolimus in healthy Chinese subjects: a population pharmacokinetic analysis.

Summary What is known and Objective: Tacrolimus (TAC) is metabolized mainly by the CYP3A subfamily and extruded into the intestine by P-glycoprotein, which is encoded by the ABCB1 gene. Several studies have suggested that the CYP3A5*3 genotype influenced the pharmacokinetics (PK) of TAC. The CYP3A4*...

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Bibliographic Details
Published in:Journal of Clinical Pharmacy & Therapeutics Vol. 36; no. 5; pp. 614 - 625
Main Authors: Shi, X.-J., Geng, F., Jiao, Z., Cui, X.-Y., Qiu, X.-Y., Zhong, M.-K.
Format: equations & formulas research tables/charts Journal Article
Published: Wiley-Blackwell Oct2011
Online Access:View this record in EBSCOhost