In vitro and in vivo anti-Helicobacter pylori activity of Calophyllum brasiliense Camb.

AIMS OF THE STUDY: Calophyllum brasiliense (Camb.) is a medicinal tree that grows particularly in the hilly and forested regions of Brazil. Preparations from its stem bark are popular remedies for the treatment of chronic ulcers. Since earlier investigations on bark extracts evidenced gastroprotecti...

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Publicado en:Journal of Ethnopharmacology Vol. 123; no. 3; pp. 452 - 459
Autores principales: Carmo Souza M, Beserra AMS, Martins DC, Villa Real V, Nunes Santos RA, Rao VS, Matos Silva R, Oliveira Martins DT
Formato: pictorial research tables/charts Journal Article
Publicado: Elsevier B.V. Jun2009
Acceso en línea:Ver este registro en EBSCOhost
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      dt: Jun2009
      vid: 123
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      pub: Elsevier B.V.
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        10.1016/j.jep.2009.03.030
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        atl: In vitro and in vivo anti-Helicobacter pylori activity of Calophyllum brasiliense Camb.
      aug:
        au:
          Carmo Souza M
          Beserra AMS
          Martins DC
          Villa Real V
          Nunes Santos RA
          Rao VS
          Matos Silva R
          Oliveira Martins DT
        affil: Department of Basic Science in Health, Faculty of Medical Science, Federal University of Mato Grosso (UFMT), Av. Fernando Correa da Costa s/n, Coxipó, Cuiabá, MT CEP: 78060-900, Brazil. macsouza@hotmail.com
      sug:
        subj:
          Helicobacter Infections Prevention and Control
          Plant Bark
          Plant Extracts Administration and Dosage
          Plant Extracts Pharmacodynamics
          Plant Stems
          Plants, Medicinal Brazil
          Alternative Therapies
          Animal Studies
          Brazil
          Descriptive Statistics
          Fisher's Exact Test
          Funding Source
          In Vitro Studies
          In Vivo Studies
          One-Way Analysis of Variance
          Post Hoc Analysis
          Rats
      ab: AIMS OF THE STUDY: Calophyllum brasiliense (Camb.) is a medicinal tree that grows particularly in the hilly and forested regions of Brazil. Preparations from its stem bark are popular remedies for the treatment of chronic ulcers. Since earlier investigations on bark extracts evidenced gastroprotective and gastric acid inhibitory properties, this study evaluated the effects of hydroethanolic extract (HEECb) and the dichloromethanic fraction (DCMF), from Calophyllum brasiliense stem bark, against Helicobacter pylori, in vitro and in vivo. MATERIALS AND METHODS: The in vitro assays were performed using the disk diffusion and broth microdilution methods to determine the minimum inhibitory concentration (MIC) values. The test substances were evaluated in vivo taking into account the delay in the gastric ulcer healing in Wistar rats, infected with Helicobacter pylori. RESULTS: DCMF appeared the most active and potent in vitro against Helicobacter pylori growth with an MIC of 31 microg/mL. In the in vivo assays, rats ulcerated by acetic acid, and inoculated with Helicobacter pylori showed a marked delay in ulcer healing. Treatment with HEECb (50, 100 and 200 mg/kg) and DCMF (100 and 200 mg/kg) reduced the ulcerated area in a dose-dependent manner. While DCMF, at 200 mg/kg, increased the prostaglandin E2 (PGE2) level, both HEECb and DCMF decreased the number of urease-positive animals, as confirmed by the reduction of Helicobacter pylori presence in histopathological analysis. CONCLUSION: The results suggest that the antiulcer activity of Calophyllum brasiliense is due, in part, to its anti-Helicobacter pylori action, validating the popular use of this species.
      pubtype: Academic Journal
      doctype:
        pictorial
        research
        tables/charts
        Journal Article
      ougenre: Article
    language: English
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