Amlodipine Ameliorates Ischemia-Induced Neovascularization in Diabetic Rats through Endothelial Progenitor Cell Mobilization.

Objectives. We investigated whether amlodipine could improve angiogenic responses in a diabetic rat model of acute myocardial infarction (AMI) through improving bone marrow endothelial progenitor cell (EPC) mobilization, in the same way as angiotensin converting enzyme inhibitors. Methods. After ind...

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Publicado en:BioMed Research International Vol. 2016; pp. 1 - 14
Autores principales: Sun, Jiayin, Xie, Jun, Kang, Lina, Ferro, Albert, Dong, Li, Xu, Biao
Formato: diagnostic images pictorial research tables/charts Journal Article
Publicado: Wiley-Blackwell 5/8/2016
Acceso en línea:Ver este registro en EBSCOhost
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      dt: 5/8/2016
      vid: 2016
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      pub: Wiley-Blackwell
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        10.1155/2016/3182764
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        atl: Amlodipine Ameliorates Ischemia-Induced Neovascularization in Diabetic Rats through Endothelial Progenitor Cell Mobilization.
      aug:
        au:
          Sun, Jiayin
          Xie, Jun
          Kang, Lina
          Ferro, Albert
          Dong, Li
          Xu, Biao
        affil: Department of Cardiology, Beijing Anzhen Hospital, Capital Medical University, Beijing 100029, China
      sug:
        subj:
          Amlodipine Administration and Dosage
          Neovascularization, Pathologic Drug Therapy
          Diabetes Mellitus Complications
          Stem Cells
          Cell Movement
          Endothelium
          Myocardial Infarction Complications
          Neovascularization, Physiologic Drug Effects
          Signal Transduction Drug Effects
          Animal Studies
          Rats
          Models, Biological
          Random Assignment
          Perindopril Administration and Dosage
          Pretest-Posttest Design
          Heart Physiology
          Ventricular Remodeling Drug Effects
          Fibrosis
          Apoptosis Drug Effects
          Vascular Endothelial Growth Factors Drug Effects
          Oxidoreductases Drug Effects
          Protein Kinases Drug Effects
          Echocardiography
          Biological Assay
          Blotting, Western
          Descriptive Statistics
          T-Tests
          One-Way Analysis of Variance
          Post Hoc Analysis
          Data Analysis Software
          P-Value
          Flow Cytometry
          Reverse Transcriptase Polymerase Chain Reaction
          Funding Source
      ab: Objectives. We investigated whether amlodipine could improve angiogenic responses in a diabetic rat model of acute myocardial infarction (AMI) through improving bone marrow endothelial progenitor cell (EPC) mobilization, in the same way as angiotensin converting enzyme inhibitors. Methods. After induction of AMI by coronary artery ligation, diabetic rats were randomly assigned to receive perindopril (2 mgkg−1 day−1), amlodipine (2.5 mgkg−1 day−1), or vehicle by gavage (n=20 per group). Circulating EPC counts before ligation and on days 1, 3, 5, 7, 14, and 28 after AMI were measured in each group. Microvessel density, cardiac function, and cardiac remodeling were assessed 4 weeks after treatment. The signaling pathway related to EPC mobilization was also measured. Results. Circulating EPC count in amlodipine- and perindopril-treated rats peaked at day 7, to an obvious higher level than the control group peak which was reached earlier (at day 5). Rats treated with amlodipine showed improved postischemia neovascularization and cardiac function, together with reduced cardiac remodeling, decreased interstitial fibrosis, and cardiomyocyte apoptosis. Amlodipine treatment also increased cardiac SDF-1/CXCR4 expression and gave rise to activation of VEGF/Akt/eNOS signaling in bone marrow. Conclusions. Amlodipine promotes neovascularization by improving EPC mobilization from bone marrow in diabetic rats after AMI, and activation of VEGF/Akt/eNOS signaling may in part contribute to this.
      pubtype: Academic Journal
      doctype:
        diagnostic images
        pictorial
        research
        tables/charts
        Journal Article
      ougenre: Article
    language: English
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