Effects of Rifampin on the Pharmacokinetics of a Single Dose of Istradefylline in Healthy Subjects.

Abstract: Istradefylline, a selective adenosine A2A inhibitor, is under development for the treatment of Parkinson's disease. The effect of oral steady‐state rifampin 600 mg/day, a potent cytochrome P450 (CYP) 3A4 inducer, on the disposition of a single oral dose of istradefylline 40 mg was determin...

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Detalles Bibliográficos
Publicado en:Journal of Clinical Pharmacology Vol. 58; no. 2; pp. 193 - 202
Autores principales: Mukai, Mayumi, Uchimura, Tatsuo, Zhang, Xiaoping, Greene, Douglas, Vergeire, Maria, Cantillon, Marc
Formato: research tables/charts Journal Article
Publicado: Wiley-Blackwell Feb2018
Acceso en línea:Ver este registro en EBSCOhost