Enzyme Inhibitory Kinetics and Molecular Docking Studies of Halo-Substituted Mixed Ester/Amide-Based Derivatives as Jack Bean Urease Inhibitors.

A series of halo-substituted mixed ester/amide-based analogues 4a-l have been prepared as jack bean urease inhibitor, which showed good to excellent inhibition of enzyme activity. The role of halo-substituted benzoyl moieties and alkyl substituted anilines in urease inhibitory kinetics was also inve...

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Publicado en:BioMed Research International pp. 1 - 12
Autores principales: Rashid, Muhammad, Rafique, Hummera, Roshan, Sadia, Shamas, Shazia, Iqbal, Zafar, Ashraf, Zaman, Abbas, Qamar, Hassan, Mubashir, Qureshi, Zia Ur Rahman, Asad, Muhammad Hassham Hassan Bin
Formato: pictorial research tables/charts Journal Article
Publicado: Wiley-Blackwell 12/24/2020
Acceso en línea:Ver este registro en EBSCOhost