Tirzepatide and the Cardiovascular Continuum: Metabolic, Cardiorenal and Heart Failure Evidence.

Tirzepatide is a first-in-class, once-weekly dual GIP and GLP-1 receptor agonist approved for type 2 diabetes and obesity. Given the tight link between hyperglycemia, adiposity, and cardiovascular disease, tirzepatide has rapidly gained interest as a broader cardiometabolic intervention. This narrat...

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Publicado en:Clinical Medicine Insights: Cardiology Vol. 20; pp. 1 - 11
Autores principales: Parlati, Antonio LM, Martini, Luca, Nardi, Ermanno, Carluccio, Raffaele, Parlati, Luca EP, Madaudo, Cristina, Perrone Filardi, Pasquale
Formato: pictorial review tables/charts Journal Article
Publicado: Sage Publications Inc. 6/16/2026
Acceso en línea:Ver este registro en EBSCOhost
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      dt: 6/16/2026
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        atl: Tirzepatide and the Cardiovascular Continuum: Metabolic, Cardiorenal and Heart Failure Evidence.
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          Parlati, Antonio LM
          Martini, Luca
          Nardi, Ermanno
          Carluccio, Raffaele
          Parlati, Luca EP
          Madaudo, Cristina
          Perrone Filardi, Pasquale
        affil: Department of Advanced Biomedical Sciences, Federico II University, Naples, Italy
      sug:
        subj:
          Diabetes Mellitus, Type 2 Drug Therapy
          Obesity Drug Therapy
          Glucagon-Like Peptide-1 Receptor Agonists Therapeutic Use
          Drug Evaluation
          Cardiovascular Risk Factors
          Risk Assessment
          Heart Failure Risk Factors
          Glycated Hemoglobin Drug Effects
          Weight Loss Drug Effects
          Waist Circumference
          Blood Pressure
          Triglycerides
          Biological Markers
          Inflammation
          Hyperlipidemia
          Hypertension
          Sleep Apnea, Obstructive
          Drug Tolerance
          Patient Safety
      ab: Tirzepatide is a first-in-class, once-weekly dual GIP and GLP-1 receptor agonist approved for type 2 diabetes and obesity. Given the tight link between hyperglycemia, adiposity, and cardiovascular disease, tirzepatide has rapidly gained interest as a broader cardiometabolic intervention. This narrative review summarizes mechanistic rationale and clinical evidence on cardiovascular risk-factor modification, cardiorenal signals, and outcome data. Across the SURPASS program in type 2 diabetes, tirzepatide produces large, dose-dependent reductions in HbA1c and substantial weight loss, with consistent benefits versus active comparators. In obesity, the SURMOUNT trials showed marked and durable weight reduction over long follow-up, with clinically relevant improvements in waist circumference, blood pressure, triglycerides, and inflammatory biomarkers. Beyond weight and glycaemia, available data suggest favorable effects on lipids, ambulatory blood pressure, inflammatory markers, and kidney-related endpoints in exploratory analyses. Tirzepatide also improves obstructive sleep apnea severity in adults with obesity. Regarding cardiovascular outcomes, SURPASS-CVOT supports cardiovascular safety by demonstrating noninferiority versus dulaglutide for 3-point major adverse cardiovascular events in patients with type 2 diabetes and established atherosclerotic cardiovascular disease (ASCVD). In obesity-related HFpEF, SUMMIT shows reductions in worsening heart failure (HF) events and improvements in health status, supporting a phenotype-specific role in HF. Overall, tirzepatide is emerging as a key therapeutic option for integrated cardiometabolic risk reduction, with ongoing research needed to define its incremental benefit versus established GLP-1 receptor agonists, long-term effectiveness in routine care, and optimal positioning across HF phenotypes.
      pubtype: Academic Journal
      doctype:
        pictorial
        review
        tables/charts
        Journal Article
      ougenre: Article
    language: English
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