Prescription cascades associated with acetylcholinesterase inhibitors use: a high-throughput sequence symmetry analysis.

Background Acetylcholinesterase inhibitors (AChEIs), are commonly prescribed for dementia and can cause adverse drug events that may lead to new prescriptions, known as prescription cascades. We aimed to identify potential AChEI-induced prescription cascades using high-throughput sequence symmetry a...

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Publicado en:Age & Ageing Vol. 55; no. 6; pp. 1 - 11
Autores principales: Newby, Danielle, Bobba, Sai Sumedha, Raventós, Berta, Rowlands, Elin J, Chen, Xihang, Molina-Porcel, Laura, Reyes, Carlen, Duarte-Salles, Talita, Delmestri, Antonella, Man, Wai Yi
Formato: Artículo
Publicado: Oxford University Press / USA Jun2026
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Acceso en línea:Ver este registro en EBSCOhost
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        atl: Prescription cascades associated with acetylcholinesterase inhibitors use: a high-throughput sequence symmetry analysis.
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          Newby, Danielle
          Bobba, Sai Sumedha
          Raventós, Berta
          Rowlands, Elin J
          Chen, Xihang
          Molina-Porcel, Laura
          Reyes, Carlen
          Duarte-Salles, Talita
          Delmestri, Antonella
          Man, Wai Yi
        affil:
          Health Data Sciences (HDS), Translational Sciences, Botnar Research Centre, University of Oxford, Oxford, UK
          Health System, University of Alabama at Birmingham  Birmingham, Alabama 35294, USA
          IDIAP Jordi Gol, Fundació Institut Universitari per a la recerca a l'Atenció Primària de Salut Jordi Gol i Gurina (IDIAPJGol), Barcelona, SpainErasmus MC Universitair Medisch Centrum Rotterdam, Department of Medical Informatics, Erasmus University Medical Center, Rotterdam, ZH, The Netherlands
          Biobanc de l'Hospital Clinic IDIBAPS, Neurological Tissue Bank of the Biobanc-Hospital Clinic-Fundació de Recerca Clínic Barcelona-Institut d'Investigacions Biomèdiques August Pi i Sunyer (FRCB-IDIBAPS), Barcelona, SpainIDIBAPS–Alzheimer's disease and other cognitive disorders unit, Neurology Service, Hospital Clínic, Barcelona, Spain
          Sardenya Primary Health Care Center, Equip d'Atenció Primària Barcelona Sardenya research unit- Sant Pau Research Institute (EAP Sarden), Barcelona, Spain
          IDIAP Jordi Gol, Fundació Institut Universitari per a la recerca a l'Atenció Primària de Salut Jordi Gol i Gurina (IDIAPJGol), Barcelona, SpainDepartment of Medical Informatics, Erasmus Medical Center, Rotterdam, Zuid-Holland, The Netherlands
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        United Kingdom
        Drug side effects
        Primary health care
        Drugs
        Benzodiazepines
        Donepezil
        Rivastigmine
        Risk assessment
        Pharmacology
        Drug allergy
        Diarrhea
        Adrenocortical hormones
        Steroids
        Cholinesterase inhibitors
        Research funding
        Piperidine
        Polypharmacy
        Descriptive statistics
        Tranquilizing drugs
        Respiratory diseases
        Deprescribing
        Neurological disorders
        Rhinorrhea
        Drug interactions
        Electronic health records
        Physician practice patterns
        Galanthamine
        Data analysis software
        Confidence intervals
        Drug eruptions
        Drug prescribing
        Sequence analysis
        Sensitivity & specificity (Statistics)
        Nausea
        Gastrointestinal diseases
      sug:
        subj:
          Drug side effects
          Primary health care
          Drugs
          United Kingdom
          Pharmaceuticals and pharmacy supplies merchant wholesalers
          Pharmaceutical and medicine manufacturing
          Drugs and Druggists' Sundries Merchant Wholesalers
          Medicinal and Botanical Manufacturing
          Benzodiazepines
          Donepezil
          Rivastigmine
          Risk assessment
          Pharmacology
          Drug allergy
          Diarrhea
          Adrenocortical hormones
          Steroids
          Cholinesterase inhibitors
          Research funding
          Piperidine
          Polypharmacy
          Descriptive statistics
          Tranquilizing drugs
          Respiratory diseases
          Deprescribing
          Neurological disorders
          Rhinorrhea
          Drug interactions
          Electronic health records
          Physician practice patterns
          Galanthamine
          Data analysis software
          Confidence intervals
          Drug eruptions
          Drug prescribing
          Sequence analysis
          Sensitivity & specificity (Statistics)
          Nausea
          Gastrointestinal diseases
      keyword:
        acetylcholinesterase inhibitors
        adverse drug events
        adverse effects of medication
        aged
        copyrightHolder:British Geriatrics Society
        copyrightYear:2026
        dementia
        donepezil
        galantamine
        gastrointestinal agents
        glucocorticoids
        https://dx.doi.org/10.1093/ageing/afag188
        inLanguage:en
        nervous system
        older people
        pharmacovigilance
        prescription cascade
        publisher:Oxford University Press
        rivastigmine
        sameAs:https://pubmed.ncbi.nlm.nih.gov/42341204/
        sensitivity analysis
        sequence symmetry analysis
        signal detection (psychology)
        united states social security administration
        acetylcholinesterase inhibitors
        adverse drug events
        adverse effects of medication
        aged
        copyrightHolder:British Geriatrics Society
        copyrightYear:2026
        dementia
        donepezil
        galantamine
        gastrointestinal agents
        glucocorticoids
        https://dx.doi.org/10.1093/ageing/afag188
        inLanguage:en
        nervous system
        older people
        pharmacovigilance
        prescription cascade
        publisher:Oxford University Press
        rivastigmine
        sameAs:https://pubmed.ncbi.nlm.nih.gov/42341204/
        sensitivity analysis
        sequence symmetry analysis
        signal detection (psychology)
        united states social security administration
      ab: Background Acetylcholinesterase inhibitors (AChEIs), are commonly prescribed for dementia and can cause adverse drug events that may lead to new prescriptions, known as prescription cascades. We aimed to identify potential AChEI-induced prescription cascades using high-throughput sequence symmetry analysis (SSA). Methods Patients aged ≥18 years with 365 days of prior observation initiating AChEIs (donepezil, rivastigmine, or galantamine) were identified from the Clinical Practice Research Datalink GOLD (2002–2022). We screened 510 drug classes and 1213 individual ingredients initiated within ±180 days of AChEI initiation (365 days in sensitivity analyses). Crude and adjusted sequence ratios (ASRs) were calculated, and positive signals were reviewed for clinical plausibility. Results We identified 66 155 AChEI initiators (median age 81 years [IQR 76–85]; 62.8% female). Among ATC classes and individual ingredients, 51 and 46 signals were positive with 28 (55%) and 22 (48%) classified as potential prescription cascades after review. Gastrointestinal drugs showed positive signals including antipropulsives (ASR 1.50 [99% CI 1.28–1.75]), loperamide (ASR 1.52 [1.30–1.77]) and cyclizine (ASR 2.10 [1.72–2.59]). Positive signals were also observed nervous system drugs such as benzodiazepine derivatives (ASR 1.83 [1.55–2.16]) and respiratory drugs including corticosteroids (ASR 1.66 [1.33–2.08]) and glucocorticoids (ASR 1.54 [1.30–1.83]). Most positive signals remained in sensitivity analysis. Conclusions These findings suggest potential AChEI-related prescription cascades consistent with gastrointestinal, neuropsychiatric, dermatological and respiratory adverse effects. While findings require further validation, this study demonstrates the utility of high-throughput signal detection to support pharmacovigilance in high-risk populations.
      pubtype: Academic Journal
      doctype: Article
      src: R
    language: English
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